EZSolution™ GSK343

A 10 mM (1 mg in 185 µl) solution of the EZH2 inhibitor GSK343 (Cat. No. 2281) in anhydrous DMSO.

Alternate Name/Synonyms: 1-Isopropyl-N-((6-methyl-2-oxo-4-propyl-1,2-dihydropyridin-3-yl)methyl)-6-(2-(4-methylpiperazin-1-yl)pyridine-4-yl)-1H-indazole-4-carboxamide

Appearance: Liquid

Appearance: A 10 mM solution in anhydrous DMSO

Appearance: N/A

Appearance: Yes

Peptide sequence: No

Salt Form: No

Molecular Formula: C₃₁H₃₉N₇O₂

Molecular Weight: 541.69

Cell-Permeable?: Yes

Purity: ≥99% by HPLC

Solubilities: N/A

Handling: Protect from light and moisture

Country of Origin: USA

Tag Line: A potent EZH2 inhibitor

MDL Number: N/A

PubChem CID: 71268957

SMILES: CCCC1=C(CNC(=O)C2=C3C=NN(C(C)C)C3=CC(=C2)C2=CC=NC(=C2)N2CCN(C)CC2)C(=O)NC(C)=C1

InChi: InChI=1S/C31H39N7O2/c1-6-7-23-14-21(4)35-31(40)26(23)18-33-30(39)25-15-24(16-28-27(25)19-34-38(28)20(2)3)22-8-9-32-29(17-22)37-12-10-36(5)11-13-37/h8-9,14-17,19-20H,6-7,10-13,18H2,1-5H3,(H,33,39)(H,35,40)

InChi Key: ULNXAWLQFZMIHX-UHFFFAOYSA-N

Category: Biochemicals